CAS
2108100-73-6
Formulation
A crystalline solid
Purity
≥97%
MW
359,5
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
A potent endocannabinoid uptake inhibitor (IC50s = 10 and 283 nM for AEA and 2-AG, respectively, in U937 cells); inhibits AEA uptake in FAAH-deficient HMC-1 human mast cells and Neuro2a mouse neuroblastoma cells (IC50s = 137 and 55 nM, respectively); increases AEA and 2-AG levels by 1.5-fold in mouse brain but not peripheral tissues (10 mg/kg, i.p. for seven days); induces a typical tetrad of hypothermia, catalepsy, analgesia, and hypomotility in mice
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).