SR 144528
CAY-9000491-5 5 mg
Data Sheet: 
SDS:
SDS:
CAS
192703-06-3
Formulation
A crystalline solid
Purity
≥98%
MW
476,1
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
SR 144528 is a cannabinoid 2 (CB2) receptor antagonist (Ki = 0.6 nM).{7912} It is selective for CB2 over CB1 receptors in CHO cells expressing the human receptors (Ki = 437 nM).{17199} SR 144528 reverses CP 55,940-induced inhibition of forskolin-induced adenylyl cyclase activity in CHO cells expressing human CB2 receptors (EC50 = 10 nM). SR 144528 (0.01 mg/kg) reduces paw swelling in a mouse model of carrageenan-induced paw edema.{14732}
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).
