Synonyms: [D-Ala2, Glu4]Deltorphin II|[D-Ala2]Deltorphin II|DADELT II|Tyr-D-Ala-Phe-Glu-Val-Val-Gly-NH2
Formulation
A solid
Purity
≥98%
MW
782,88328
Shipment
-20
Long Term Storage
-20
Shelf Life
4 years from production
Description
A peptide agonist of δ2-opioid receptors; selective for δ-opioid receptors over μ- and κ-opioid receptors in radioligand bindings assays (Kis = 0.0033, >1, and >1 µM, respectively); induces [35S]GTPγS binding in mouse brain membrane preparations (EC50 = 0.034 µM); decreases the infarction zone:risk zone ratio in a rat model of myocardial ischemia-reperfusion injury induced by coronary occlusion at 0.12 mg/kg; intrathecal administration increases latency to withdraw in the paw pressure and tail-flick tests in rats at 15 µg/animal
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).