CP 809,101
CAY-24214-5 5 mg
Data Sheet: 
SDS:
SDS:
CAS
479683-64-2
Formulation
A crystalline solid
Purity
≥98%
MW
304,77454
Shipment
-20
Long Term Storage
-20
Shelf Life
1460
Description
A potent 5-HT2C receptor agonist (Ki = 1.6 nM); selective for human 5-HT2C and rat 5-HT2C over human 5-HT2A, 5-HT2B, and rat 5-HT2A receptors in a FLIPR assay (EC50s = 0.11, 0.06, 153, 65.3, and 119 nM, respectively) as well as human dopamine D2, histamine H1, and α1- and α2-adrenergic receptors (Kis = 872, 828, 217, and 956 nM, respectively); inhibits the conditioned avoidance response, hyperactivity induced by PCP and D-amphetamine, and spontaneous locomotor activity in rats (ED50s = 4.8, 2.4, 2.9, and 2 mg/kg, respectively); reduces reinstatement of drug-seeking behavior in cocaine-primed rats (0.01-1 μg/0.2 μl/side in central amygdala); reduces reinstatement of food-seeking behavior in a rat model of dietary relapse
ESCLUSIVAMENTE PER USO DI RICERCA (RUO) e non per uso terapeutico o diagnostico su uomini o animali. Il prodotto NON è un Dispositivo Medico o un Diagnostico in Vitro.
PRODUCT FOR RESEARCH USE ONLY (RUO) and not for therapeutic or diagnostic use on humans or animals. The product is NOT a Medical Device or an In-Vitro Diagnostic (IVD).
